ABX Datasheet Product Number 9771

ABX advanced biochemical compounds


Catalogue Number	Product	Order number / Unit

9771	Gluc-[Lys⁰,Lys(ivDde)⁵]-TOCA	9771.0001: 1 mg per vial 9771.0010: 10 mg per vial Please inquire for customized filling and bulk quantities.
	Precursor for Gluc-Lys([¹⁸F]FP)-TOCA


	Molar Mass: 1545.82
	C₇₄H₁₀₄N₁₂O₂₀S₂
	CAS-RN not yet assigned

	Colourless to off-white freeze-dried solid packaged in screw cap vials.


	Purity: ≥ 95 %
	Certificates: CoA; MS (identity); HPLC (purity)
	Chemical Name: Sequence: (1-deoxy-D-fructosyl)-Lys-D-Phe-Cys-Tyr-D-Trp-Lys(ivDde)-Thr-Cys-Thr-OH, cyclic disulfide
	Synonymes: (N^α-(1-deoxy-D-fructosyl)-[Lys⁰-Tyr³-Lys(Dde)⁵]-octreotate; Precursor for [¹⁸F]FP-Gluc-TOCA; N-α-(1-deoxy-D-fructosyl)-KfCYw-K(ivDde)-TCT-OH, cyclic C^2,7; Gluc-Lys([¹⁸F]FP)-TOCA = N^α-(1-deoxy-D-fructosyl)-N^ε-(2-[¹⁸F]fluoropropionyl)- Lys⁰-Tyr³-octreotate
	Literature: Meisetschlaeger G. et al. Gluc-Lys([¹⁸F]FP)-TOCA PET in Patients with SSTR-Positive Tumors: Biodistribution and Diagnostic Evaluation Compared with [¹¹¹In]DTPA-Octreotide. J. Nucl. Med. 2006, 47, 566-573.
	Vaidyanathan G. et al. Synthesis and Evaluation of Glycosylated Octreotate Analogues Labeled with Radioiodine and ²¹¹At via a Tin Precursor. Bioconjugate Chem. 2006, 17, 195-203.



	date of product catalogue issue: 10 May 2017